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Discovery of novel TASK-3 channel blockers using a pharmacophore-based virtual screening
Fecha de emisión
2019
Autor(es)
Ramírez D.
Concha G.
Arévalo B.
Prent-Peñaloza L.
Zúñiga L.
Kiper A.K.
Rinné S.
Reyes-Parada M.
Decher N.
González W.
Caballero J.
DOI
10.3390/ijms20164014
Temas
Drug design
Lead optimization
Pharmacophore-based v...
TASK channels blocker...
TASK-3 channel
potassium channel blo...
KCNK9 protein, human
potassium channel blo...
tandem pore domain po...
Article
binding site
carbon nuclear magnet...
controlled study
crystal structure
Fourier transform inf...
high throughput scree...
human
human cell
hydrogen bond
mass spectrometry
molecular docking
molecular dynamics
patch clamp technique...
pharmacophore
protein conformation
protein expression
proton nuclear magnet...
stereochemistry
drug design
HEK293 cell line
molecular docking
Drug Design
HEK293 Cells
Humans
Molecular Docking Sim...
Potassium Channel Blo...
Potassium Channels, T...
Archivo(s)